Crystal structure of T2R-TTL-PM534 complex
收藏Protein Data Bank Japan2026-03-04 更新2026-04-19 收录
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Crystal structure of T2R-TTL-PM534 complex Descriptor: (4R)-N-[(1R)-1-[4-(cyclopropylmethoxy)-6-oxidanylidene-pyran-2-yl]butyl]-4-methyl-2-[(E)-C-methyl-N-oxidanyl-carbonimidoyl]-5H-1,3-thiazole-4-carboxamide, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CALCIUM ION, ... Authors: Oliva, M.A, Diaz, J.F, Cuevas, C. Deposit date: 2022-05-25 Release date: 2023-11-29 Last modified: 2026-03-04 Method: X-RAY DIFFRACTION (2.45 Å) Cite: PM534, an Optimized Target-Protein Interaction Strategy through the Colchicine Site of Tubulin. J.Med.Chem., 67, 2024
创建时间:
2022-05-25



