five

Crystal structure of LSD1 in complex with compound 5

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Protein Data Bank Japan2023-11-29 更新2026-04-25 收录
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Crystal structure of LSD1 in complex with compound 5 Descriptor: 3-[3,5-bis(fluoranyl)-2-[(2-fluoranylpyridin-4-yl)methoxy]phenyl]propanal, FLAVIN-ADENINE DINUCLEOTIDE, GLYCEROL, ... Authors: Niwa, H, Koda, Y, Sato, S, Yamamoto, H, Koyama, H, Umehara, T. Deposit date: 2021-10-20 Release date: 2022-06-01 Last modified: 2023-11-29 Method: X-RAY DIFFRACTION (2.91 Å) Cite: Design and Synthesis of Tranylcypromine-Derived LSD1 Inhibitors with Improved hERG and Microsomal Stability Profiles. Acs Med.Chem.Lett., 13, 2022
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2021-10-20
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