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Crystal structure of BRDT bromodomain 2 in complex with CDD-1102

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Protein Data Bank Japan2023-10-18 更新2026-03-21 收录
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Crystal structure of BRDT bromodomain 2 in complex with CDD-1102 Descriptor: BETA-MERCAPTOETHANOL, Bromodomain testis-specific protein, N~1~-(5-{[3-(4-amino-2-methylphenyl)-1-methyl-1H-indazole-5-carbonyl]amino}-2-methylphenyl)-N~4~-methylbenzene-1,4-dicarboxamide Authors: Sharma, R, Kaur, G, Yu, Z, Ku, A.F, Anglin, J.L, Ucisik, M.N, Faver, J.C, Sankaran, B, Kim, C, Matzuk, M.M. Deposit date: 2021-01-03 Release date: 2021-06-30 Last modified: 2023-10-18 Method: X-RAY DIFFRACTION (2.27 Å) Cite: Discovery and characterization of bromodomain 2-specific inhibitors of BRDT. Proc.Natl.Acad.Sci.USA, 118, 2021
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2021-01-03
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