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Human EphA3 Kinase domain in complex with ligand 66

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Protein Data Bank Japan2023-11-08 更新2026-03-21 收录
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Human EphA3 Kinase domain in complex with ligand 66 Descriptor: 7-(5-hydroxy-2-methylphenyl)-8-(2-methoxyphenyl)-1-methyl-1H-imidazo[2,1-f]purine-2,4(3H,8H)-dione, EPH receptor A3 Authors: Dong, J, Caflisch, A. Deposit date: 2012-08-10 Release date: 2013-01-23 Last modified: 2023-11-08 Method: X-RAY DIFFRACTION (2.195 Å) Cite: Optimization of Inhibitors of the Tyrosine Kinase EphB4. 2. Cellular Potency Improvement and Binding Mode Validation by X-ray Crystallography. J.Med.Chem., 56, 2013
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2012-08-10
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