Co-crystal Structure of JNK1 and AX13587
收藏Protein Data Bank Japan2024-02-28 更新2026-03-21 收录
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Co-crystal Structure of JNK1 and AX13587 Descriptor: Mitogen-activated protein kinase 8, N-[1-(4-fluorophenyl)cyclopropyl]-4-[(trans-4-hydroxycyclohexyl)amino]imidazo[1,2-a]quinoxaline-8-carboxamide Authors: Walter, R.L, Ranieri, G.M, Riggs, A.M, Weissig, H, Li, B, Shreder, K.R. Deposit date: 2013-06-13 Release date: 2013-08-21 Last modified: 2024-02-28 Method: X-RAY DIFFRACTION (1.95 Å) Cite: Hit-to-lead optimization and kinase selectivity of imidazo[1,2-a]quinoxalin-4-amine derived JNK1 inhibitors. Bioorg.Med.Chem.Lett., 23, 2013
创建时间:
2013-06-13



