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1.68A STRUCTURE PCAF BROMODOMAIN WITH 4-chloro-2-methyl-5-(methylamino)pyridazin-3(2H)-one

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Protein Data Bank Japan2024-06-19 更新2026-03-21 收录
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https://pdbj.org/mine/summary/5mkx
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1.68A STRUCTURE PCAF BROMODOMAIN WITH 4-chloro-2-methyl-5-(methylamino)pyridazin-3(2H)-one Descriptor: 1,4-BUTANEDIOL, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, 4-chloranyl-2-methyl-5-(methylamino)pyridazin-3-one, ... Authors: Chung, C.-W. Deposit date: 2016-12-05 Release date: 2017-12-20 Last modified: 2024-06-19 Method: X-RAY DIFFRACTION (1.68 Å) Cite: Discovery of a Potent, Cell Penetrant, and Selective p300/CBP-Associated Factor (PCAF)/General Control Nonderepressible 5 (GCN5) Bromodomain Chemical Probe. J. Med. Chem., 60, 2017
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2016-12-05
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