Human artd1 (parp1) - catalytic domain in complex with inhibitor xav939
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https://pdbj.org/mine/summary/4r5w
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Human artd1 (parp1) - catalytic domain in complex with inhibitor xav939 Descriptor: 2-[4-(trifluoromethyl)phenyl]-7,8-dihydro-5H-thiopyrano[4,3-d]pyrimidin-4-ol, Poly [ADP-ribose] polymerase 1, SULFATE ION Authors: Karlberg, T, Thorsell, A.G, Schuler, H. Deposit date: 2014-08-22 Release date: 2015-09-02 Last modified: 2023-09-20 Method: X-RAY DIFFRACTION (2.84 Å) Cite: Structural Basis for Potency and Promiscuity in Poly(ADP-ribose) Polymerase (PARP) and Tankyrase Inhibitors. J.Med.Chem., 60, 2017
创建时间:
2014-08-22



