Structure of TTBK1 kinase domain in complex with Compound 18
收藏Protein Data Bank Japan2023-10-18 更新2026-03-21 收录
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Structure of TTBK1 kinase domain in complex with Compound 18 Descriptor: (3S)-1-[1-(2-aminopyrimidin-4-yl)-1H-pyrazolo[4,3-c]pyridin-6-yl]-3-methylpent-1-yn-3-ol, Tau-tubulin kinase 1 Authors: Chodaprambil, J.V. Deposit date: 2020-08-28 Release date: 2021-05-19 Last modified: 2023-10-18 Method: X-RAY DIFFRACTION (2.15 Å) Cite: Discovery of Potent and Brain-Penetrant Tau Tubulin Kinase 1 (TTBK1) Inhibitors that Lower Tau Phosphorylation In Vivo. J.Med.Chem., 64, 2021
创建时间:
2020-08-28



