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JAK2 kinase (JH1 domain) in complex with 2,6-DICHLORO-N-{2-[(CYCLOPROPYLCARBONYL)AMINO]PYRIDIN-4-YL}BENZAMIDE

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Protein Data Bank Japan2024-11-20 更新2026-03-21 收录
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https://pdbj.org/mine/summary/4gmy
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JAK2 kinase (JH1 domain) in complex with 2,6-DICHLORO-N-{2-[(CYCLOPROPYLCARBONYL)AMINO]PYRIDIN-4-YL}BENZAMIDE Descriptor: 2,6-dichloro-N-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}benzamide, Tyrosine-protein kinase JAK2 Authors: Murray, J.M, Shia, S. Deposit date: 2012-08-16 Release date: 2013-06-19 Last modified: 2024-11-20 Method: X-RAY DIFFRACTION (2.403 Å) Cite: Lead identification of novel and selective TYK2 inhibitors. Eur.J.Med.Chem., 67, 2013
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2012-08-16
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