Human MST3 (STK24) kinase in complex with inhibitor MR24
收藏Protein Data Bank Japan2024-06-19 更新2026-04-19 收录
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https://pdbj.org/mine/summary/8qlr
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Human MST3 (STK24) kinase in complex with inhibitor MR24 Descriptor: 1,2-ETHANEDIOL, 8-(4-azanylbutyl)-2-[1,3-bis(oxidanyl)propan-2-ylamino]-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]pyrido[2,3-d]pyrimidin-7-one, Serine/threonine-protein kinase 24 Authors: Balourdas, D.I, Rak, M, Knapp, S, Joerger, A.C, Structural Genomics Consortium (SGC) Deposit date: 2023-09-20 Release date: 2023-11-08 Last modified: 2024-06-19 Method: X-RAY DIFFRACTION (1.85 Å) Cite: Development of Selective Pyrido[2,3- d ]pyrimidin-7(8 H )-one-Based Mammalian STE20-Like (MST3/4) Kinase Inhibitors. J.Med.Chem., 67, 2024
创建时间:
2023-09-20



