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Rat branched chain ketoacid dehydrogenase kinase in complex with inhibitor

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Protein Data Bank Japan2025-02-26 更新2026-05-24 收录
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Rat branched chain ketoacid dehydrogenase kinase in complex with inhibitor Descriptor: (3M)-6-fluoro-3-(2,4,5-trifluoro-3-methoxyphenyl)-1-benzothiophene-2-carboxylic acid, ADENOSINE-5'-DIPHOSPHATE, Branched-chain alpha-ketoacid dehydrogenase kinase, ... Authors: Liu, S. Deposit date: 2024-09-05 Release date: 2024-11-27 Last modified: 2025-02-26 Method: X-RAY DIFFRACTION (2.155 Å) Cite: Discovery of First Branched-Chain Ketoacid Dehydrogenase Kinase (BDK) Inhibitor Clinical Candidate PF-07328948. J.Med.Chem., 68, 2025

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2024-09-05
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