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Aurora A kinase in complex with TPX2-inhibitor 3

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Protein Data Bank Japan2024-09-25 更新2026-05-23 收录
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Aurora A kinase in complex with TPX2-inhibitor 3 Descriptor: (1~{R},2~{R})-cyclohexane-1,2-dicarboxylic acid, 4-(4-chlorophenyl)-1~{H}-indole-6-carboxylic acid, ACETATE ION, ... Authors: Fischer, G, Rocaboy, M, Blaszczyk, B, Moschetti, T, Wang, X, Scott, D.E, Coyne, A.G, Dagostin, C, Rooney, T, Bayly, A, Feng, J, Asteian, A, Alcaide-Lopez, A, Stockwell, S, Skidmore, J, Venkitaraman, A.R, Abell, C, Blundell, T.L, Hyvonen, M. Deposit date: 2022-12-20 Release date: 2024-01-10 Last modified: 2024-09-25 Method: X-RAY DIFFRACTION (2.41 Å) Cite: Selective Aurora A-TPX2 Interaction Inhibitors Have In Vivo Efficacy as Targeted Antimitotic Agents. J.Med.Chem., 67, 2024

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2022-12-20
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