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Crystal structure of IRAK4 kinase domain with compound 4

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Protein Data Bank Japan2024-11-06 更新2026-05-23 收录
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Crystal structure of IRAK4 kinase domain with compound 4 Descriptor: CHLORIDE ION, GLYCEROL, Interleukin-1 receptor-associated kinase 4, ... Authors: Weiss, M.M, Zheng, X, Browne, C.M, Campbell, V, Chen, D, Enerson, B, Fei, X, Huang, X, Klaus, C.R, Li, H, Mayo, M, McDonald, A.A, Paul, A, Sharma, K, Shi, Y, Slavin, A, Walter, D.M, Yuan, K, Zhang, Y, Zhu, X, Kelleher, J, Ji, N, Walker, D, Mainolfi, N. Deposit date: 2023-11-21 Release date: 2024-07-03 Last modified: 2024-11-06 Method: X-RAY DIFFRACTION (2.92 Å) Cite: Discovery of KT-413, a Targeted Protein Degrader of IRAK4 and IMiD Substrates Targeting MYD88 Mutant Diffuse Large B-Cell Lymphoma. J.Med.Chem., 67, 2024

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2023-11-21
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