Aurora A in complex with ATP and AA35.
收藏Protein Data Bank Japan2024-10-16 更新2026-03-21 收录
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Aurora A in complex with ATP and AA35. Descriptor: 2-(3-bromophenyl)-8-fluoroquinoline-4-carboxylic acid, ADENOSINE-5'-TRIPHOSPHATE, Aurora kinase A, ... Authors: Janecek, M, Rossmann, M, Sharma, P, Emery, A, McKenzie, G, Huggins, D, Stockwell, S, Stokes, J.A, Almeida, E.G, Hardwick, B, Narvaez, A.J, Hyvonen, M, Spring, D.R, Venkitaraman, A. Deposit date: 2015-09-09 Release date: 2016-07-20 Last modified: 2024-10-16 Method: X-RAY DIFFRACTION (2.05 Å) Cite: Allosteric modulation of AURKA kinase activity by a small-molecule inhibitor of its protein-protein interaction with TPX2. Sci Rep, 6, 2016
创建时间:
2015-09-09



