遇见数据集

C-TERMINAL BROMODOMAIN OF HUMAN BRD2 WITH 7,8-dimethoxy-3-methyl-1,3-dihydro-2H-benzo[d]azepin-2-one

收藏
Protein Data Bank Japan2024-05-01 更新2026-05-23 收录
数据链接:
官方服务:

资源简介:

C-TERMINAL BROMODOMAIN OF HUMAN BRD2 WITH 7,8-dimethoxy-3-methyl-1,3-dihydro-2H-benzo[d]azepin-2-one Descriptor: 1,2-ETHANEDIOL, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 7,8-dimethoxy-3-methyl-1~{H}-3-benzazepin-2-one, ... Authors: Chung, C. Deposit date: 2022-09-22 Release date: 2022-11-30 Last modified: 2024-05-01 Method: X-RAY DIFFRACTION (1.619 Å) Cite: Identification and Optimization of a Ligand-Efficient Benzoazepinone Bromodomain and Extra Terminal (BET) Family Acetyl-Lysine Mimetic into the Oral Candidate Quality Molecule I-BET432. J.Med.Chem., 65, 2022

创建时间:
2022-09-22
二维码
社区交流群
二维码
科研交流群
商业服务