five

Crystal Structure of Bovine G Protein Coupled-Receptor Kinase 5 in Complex with CCG215022

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Protein Data Bank Japan2023-09-27 更新2026-03-21 收录
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Crystal Structure of Bovine G Protein Coupled-Receptor Kinase 5 in Complex with CCG215022 Descriptor: (4S)-4-{4-fluoro-3-[(pyridin-2-ylmethyl)carbamoyl]phenyl}-N-(1H-indazol-5-yl)-6-methyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide, G protein-coupled receptor kinase 5, SULFATE ION Authors: Homan, K.T, Tesmer, J.J.G. Deposit date: 2014-10-13 Release date: 2015-06-10 Last modified: 2023-09-27 Method: X-RAY DIFFRACTION (2.42 Å) Cite: Crystal Structure of G Protein-coupled Receptor Kinase 5 in Complex with a Rationally Designed Inhibitor. J.Biol.Chem., 290, 2015
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2014-10-13
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