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Crystal structure of acetyltransferase Eis from Mycobacterium tuberculosis in complex with haloperidol

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Protein Data Bank Japan2023-10-18 更新2026-03-21 收录
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Crystal structure of acetyltransferase Eis from Mycobacterium tuberculosis in complex with haloperidol Descriptor: 4-[4-(4-chlorophenyl)-4-hydroxypiperidin-1-yl]-1-(4-fluorophenyl)butan-1-one, CHLORIDE ION, GLYCEROL, ... Authors: Punetha, A, Garneau-Tsodikova, S, Tsodikov, O.V. Deposit date: 2020-05-17 Release date: 2021-06-02 Last modified: 2023-10-18 Method: X-RAY DIFFRACTION (2.03 Å) Cite: Structure-based design of haloperidol analogues as inhibitors of acetyltransferase Eis from Mycobacterium tuberculosis to overcome kanamycin resistance Rsc Med Chem, 12, 2021
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2020-05-17
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