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Anaplastic Lymphoma Kinase with a novel carboline inhibitor

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Protein Data Bank Japan2024-01-31 更新2026-05-23 收录
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Anaplastic Lymphoma Kinase with a novel carboline inhibitor Descriptor: 3-(dimethylamino)-1-[3-[4-(4-methylpiperazin-1-yl)phenyl]-9~{H}-pyrido[2,3-b]indol-6-yl]prop-2-en-1-one, ALK tyrosine kinase receptor Authors: Mologni, L, Scapozza, L, Gambacorti-Passerini, C, Tardy, S, Goekjian, P, Robinson, C, Brown, D. Deposit date: 2022-08-17 Release date: 2022-09-14 Last modified: 2024-01-31 Method: X-RAY DIFFRACTION (1.645 Å) Cite: Discovery of Novel alpha-Carboline Inhibitors of the Anaplastic Lymphoma Kinase. Acs Omega, 7, 2022

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2022-08-17
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