five

Structure of phosphorylated Thr160 CDK2/cyclin A in complex with the inhibitor meriolin 5

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Protein Data Bank Japan2024-10-30 更新2026-03-21 收录
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Structure of phosphorylated Thr160 CDK2/cyclin A in complex with the inhibitor meriolin 5 Descriptor: 4-(4-propoxy-1H-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amine, Cell division protein kinase 2, Cyclin-A2, ... Authors: Echalier, A, Bettayeb, K, Ferandin, Y, Lozach, O, Clement, M, Valette, A, Liger, F, Marquet, B, Morris, J.C, Endicott, J.A, Joseph, B, Meijer, L. Deposit date: 2007-11-29 Release date: 2008-02-12 Last modified: 2024-10-30 Method: X-RAY DIFFRACTION (2.3 Å) Cite: Meriolins, a new class of cell death inducing kinase inhibitors with enhanced selectivity for cyclin-dependent kinases Cancer Res., 67, 2007
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2007-11-29
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