Lewis Acid and (Hypo)iodite Relay Catalysis Allows a Strategy for the Synthesis of Polysubstituted Azetidines and Tetrahydroquinolines
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https://figshare.com/articles/dataset/Lewis_Acid_and_Hypo_iodite_Relay_Catalysis_Allows_a_Strategy_for_the_Synthesis_of_Polysubstituted_Azetidines_and_Tetrahydroquinolines/4003983
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资源简介：
A catalytic [3 + 1]-annulation reaction
between cyclopropane 1,1-diester
and aromatic amine is developed based on the relay catalysis strategy.
Lewis acid-catalyzed nucleophilic ring opening of cyclopropane 1,1-diester
with aromatic amine and (hypo)iodite-catalyzed C–N bond formation
are combined successfully in one reaction. Using this reaction, biologically
important azetidines and tetrahydroquinolines can be prepared directly.
创建时间：
2016-10-17
