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Crystal structure of 2-(3-alkoxy-1-azetidinyl) quinolines as PDE10A Inhibitors

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Protein Data Bank Japan2024-11-13 更新2026-03-21 收录
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Crystal structure of 2-(3-alkoxy-1-azetidinyl) quinolines as PDE10A Inhibitors Descriptor: GLYCEROL, SULFATE ION, ZINC ION, ... Authors: Chmait, S. Deposit date: 2014-06-08 Release date: 2014-12-17 Last modified: 2024-11-13 Method: X-RAY DIFFRACTION (2.77 Å) Cite: Synthesis and preliminary biological evaluation of potent and selective 2-(3-alkoxy-1-azetidinyl) quinolines as novel PDE10A inhibitors with improved solubility. Bioorg.Med.Chem., 22, 2014

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2014-06-08
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