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RIP2 Kinase Catalytic Domain (1 - 310) complex with Biphenylsulfonamide

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Protein Data Bank Japan2024-01-10 更新2026-03-21 收录
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RIP2 Kinase Catalytic Domain (1 - 310) complex with Biphenylsulfonamide Descriptor: 2,6-bis(fluoranyl)-N-[3-[5-[2-[(3-methylsulfonylphenyl)amino]pyrimidin-4-yl]-2-morpholin-4-yl-1,3-thiazol-4-yl]phenyl]benzenesulfonamide, RECEPTOR-INTERACTING SERINE/THREONINE-PROTEIN KINASE 2 Authors: Charnley, A.K, Convery, M.A, Lakdawala Shah, A, Jones, E, Hardwicke, P, Bridges, A, Votta, B.J, Gough, P.J, Marquis, R.W, Bertin, J, Casillas, L. Deposit date: 2015-09-24 Release date: 2015-10-21 Last modified: 2024-01-10 Method: X-RAY DIFFRACTION (2.79 Å) Cite: Crystal Structures of Human Rip2 Kinase Catalytic Domain Complexed with ATP-Competitive Inhibitors: Foundations for Understanding Inhibitor Selectivity. Bioorg.Med.Chem., 23, 2015

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2015-09-24
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