Structure of Plasmodium falciparum 20S proteasome with bound bortezomib

Structure of Plasmodium falciparum 20S proteasome with bound bortezomib Descriptor: 20S proteasome alpha-1 subunit, 20S proteasome alpha-2 subunit, 20S proteasome alpha-3 subunit, ... Authors: Morton, C.J, Metcalfe, R.D, Liu, B, Xie, S.C, Hanssen, E, Leis, A.P, Tilley, L, Griffin, M.D.W. Deposit date: 2021-03-05 Release date: 2021-09-22 Last modified: 2025-06-04 Method: ELECTRON MICROSCOPY (3.4 Å) Cite: Design of proteasome inhibitors with oral efficacy in vivo against Plasmodium falciparum and selectivity over the human proteasome. Proc.Natl.Acad.Sci.USA, 118, 2021