five

Crystal structure of BRD2 second bromodomain in complex with SGC-CBP30 chemical probe

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Protein Data Bank Japan2024-05-08 更新2026-03-21 收录
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Crystal structure of BRD2 second bromodomain in complex with SGC-CBP30 chemical probe Descriptor: 1,2-ETHANEDIOL, 2-[2-(3-chloro-4-methoxyphenyl)ethyl]-5-(3,5-dimethyl-1,2-oxazol-4-yl)-1-[(2S)-2-(morpholin-4-yl)propyl]-1H-benzimidazole, Bromodomain-containing protein 2 Authors: Tallant, C, Hay, D, Krojer, T, Nunez-Alonso, G, Picaud, S, Newman, J.A, Fedorov, O, von Delft, F, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Brennan, P.E, Knapp, S, Structural Genomics Consortium (SGC) Deposit date: 2015-06-02 Release date: 2015-07-01 Last modified: 2024-05-08 Method: X-RAY DIFFRACTION (1.4 Å) Cite: Crystal structure of BRD2 second bromodomain in complex with a 3,5-dimethylisoxazol ligand To Be Published
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2015-06-02
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