Crystal structure of the human BRPF1 bromodomain in complex with BZ073
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Crystal structure of the human BRPF1 bromodomain in complex with BZ073 Descriptor: Peregrin, ~{N}-[1,4-diethyl-2,3-bis(oxidanylidene)-7-piperidin-1-yl-quinoxalin-6-yl]-2-(4-methylpiperazin-1-yl)ethanamide Authors: Zhu, J, Caflisch, A. Deposit date: 2017-01-20 Release date: 2018-02-14 Last modified: 2024-05-08 Method: X-RAY DIFFRACTION (1.25 Å) Cite: Structure-based discovery of selective BRPF1 bromodomain inhibitors. Eur J Med Chem, 155, 2018
创建时间:
2017-01-20



