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Strategic design of catalytic lysine-targeting reversible covalent BCR-ABL Inhibitors

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Protein Data Bank Japan2024-10-23 更新2026-03-21 收录
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Strategic design of catalytic lysine-targeting reversible covalent BCR-ABL Inhibitors Descriptor: Tyrosine-protein kinase ABL1, [4-[5-[5-(dimethylcarbamoyl)pyridin-3-yl]-1H-pyrrolo[2,3-b]pyridin-3-yl]-2-methyl-phenyl]boronic acid Authors: Anantharajan, J, Baburajendran, N. Deposit date: 2020-06-16 Release date: 2021-06-09 Last modified: 2024-10-23 Method: X-RAY DIFFRACTION (2.723 Å) Cite: Strategic Design of Catalytic Lysine-Targeting Reversible Covalent BCR-ABL Inhibitors*. Angew.Chem.Int.Ed.Engl., 60, 2021

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2020-06-16
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