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CRYSTAL STRUCTURE OF THE FIRST BROMODOMAIN OF HUMAN BRD4 IN COMPLEX WITH DB-1-264-2

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Protein Data Bank Japan2023-09-27 更新2026-03-21 收录
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CRYSTAL STRUCTURE OF THE FIRST BROMODOMAIN OF HUMAN BRD4 IN COMPLEX WITH DB-1-264-2 Descriptor: 1,2-ETHANEDIOL, 4-[[(7~{R})-8-cyclopentyl-7-ethyl-5-methyl-6-oxidanylidene-7~{H}-pteridin-2-yl]-methyl-amino]-3-methoxy-~{N}-(1-methylpiperidin-4-yl)benzamide, Bromodomain-containing protein 4 Authors: Zhu, J.-Y, Ember, S.W, Schonbrunn, E. Deposit date: 2016-06-17 Release date: 2017-08-09 Last modified: 2023-09-27 Method: X-RAY DIFFRACTION (1.51 Å) Cite: Assessment of Bromodomain Target Engagement by a Series of BI2536 Analogues with Miniaturized BET-BRET. ChemMedChem, 11, 2016
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2016-06-17
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