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Inhibitors of Jak2 Kinase domain

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Protein Data Bank Japan2023-12-20 更新2026-03-21 收录
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Inhibitors of Jak2 Kinase domain Descriptor: 5-FLUORO-4-[(1S)-1-(5-FLUOROPYRIMIDIN-2-YL)ETHOXY]-N-(5-METHYL-1H-PYRAZOL-3-YL)-6-MORPHOLINO-PYRIMIDIN-2-AMINE, ACETYL GROUP, TYROSINE-PROTEIN KINASE JAK2 Authors: Read, J, Green, I, Pollard, H, Howard, T, Mott, R. Deposit date: 2013-02-11 Release date: 2013-04-17 Last modified: 2023-12-20 Method: X-RAY DIFFRACTION (2.51 Å) Cite: Discovery of Novel Jak2-Stat Pathway Inhibitors with Extended Residence Time on Target. Bioorg.Med.Chem.Lett., 23, 2013

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2013-02-11
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