Crystal Structure of SETD2 Bound to an Indole-based Inhibitor
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Crystal Structure of SETD2 Bound to an Indole-based Inhibitor Descriptor: Histone-lysine N-methyltransferase SETD2, N-[(1R,3S)-3-(4-acetylpiperazin-1-yl)cyclohexyl]-4-fluoro-7-methyl-1H-indole-2-carboxamide, S-ADENOSYLMETHIONINE, ... Authors: Farrow, N.A. Deposit date: 2022-02-11 Release date: 2022-08-31 Last modified: 2024-04-03 Method: X-RAY DIFFRACTION (2.438 Å) Cite: Conformational-Design-Driven Discovery of EZM0414: A Selective, Potent SETD2 Inhibitor for Clinical Studies. Acs Med.Chem.Lett., 13, 2022
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2022-02-11
