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Human GKRP bound to AMG-0265 (N-[(R)-(2-CHLOROPHENYL){7-[4-(2-HYDROXYPROPAN-2-YL) PYRIDIN-2-YL]-1-BENZOTHIOPHEN-2-YL}METHYL]CYCLOPROPANESULFONAMIDE) and Sorbitol-6-phosphate

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Protein Data Bank Japan2023-09-20 更新2026-03-21 收录
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https://pdbj.org/mine/summary/4pxs
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Human GKRP bound to AMG-0265 (N-[(R)-(2-CHLOROPHENYL){7-[4-(2-HYDROXYPROPAN-2-YL) PYRIDIN-2-YL]-1-BENZOTHIOPHEN-2-YL}METHYL]CYCLOPROPANESULFONAMIDE) and Sorbitol-6-phosphate Descriptor: D-SORBITOL-6-PHOSPHATE, GLYCEROL, Glucokinase regulatory protein, ... Authors: Jordan, S.R, Chmait, S. Deposit date: 2014-03-24 Release date: 2015-03-18 Last modified: 2023-09-20 Method: X-RAY DIFFRACTION (2.6 Å) Cite: Discovery and Structure-Guided Optimization of Diarylmethanesulfonamide Disruptors of GK-GKRP Binding. To be Published
创建时间:
2014-03-24
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