Crystal structure of the first bromodomain of human BRD4 in complex with SJ001011461-1
收藏Protein Data Bank Japan2023-10-18 更新2026-04-19 收录
下载链接：
https://pdbj.org/mine/summary/7rmd
下载链接
链接失效反馈官方服务：
资源简介：
Crystal structure of the first bromodomain of human BRD4 in complex with SJ001011461-1 Descriptor: 1,2-ETHANEDIOL, 2-[(6S,10R)-4-(4-chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl]-N-(1,3,4-thiadiazol-2-yl)acetamide, Bromodomain-containing protein 4 Authors: Stachowski, T.R, Fischer, M. Deposit date: 2021-07-27 Release date: 2022-08-03 Last modified: 2023-10-18 Method: X-RAY DIFFRACTION (1.18 Å) Cite: From PROTAC to inhibitor: Structure-guided discovery of potent and orally bioavailable BET inhibitors. Eur.J.Med.Chem., 251, 2023
创建时间：
2021-07-27
