Crystal structure of TL11-128 bound to TAK1-TAB1
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Crystal structure of TL11-128 bound to TAK1-TAB1 Descriptor: Mitogen-activated protein kinase kinase kinase 7,TGF-beta-activated kinase 1 and MAP3K7-binding protein 1, ~{N}-[2-[5-chloranyl-2-[(1-methylpyrazol-4-yl)amino]pyrimidin-4-yl]oxyphenyl]prop-2-enamide Authors: Gurbani, D, Westover, K.D. Deposit date: 2016-04-25 Release date: 2017-02-15 Last modified: 2024-10-16 Method: X-RAY DIFFRACTION (2.371 Å) Cite: Structure-guided development of covalent TAK1 inhibitors. Bioorg. Med. Chem., 25, 2017
创建时间:
2016-04-25



