遇见数据集

BRD2_Bromodomain1 complex with inhibitor 744

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Protein Data Bank Japan2024-03-13 更新2026-03-21 收录
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BRD2_Bromodomain1 complex with inhibitor 744 Descriptor: 1,2-ETHANEDIOL, Bromodomain-containing protein 2, N-ethyl-4-[2-(4-fluoro-2,6-dimethylphenoxy)-5-(2-hydroxypropan-2-yl)phenyl]-6-methyl-7-oxo-6,7-dihydro-1H-pyrrolo[2,3-c]pyridine-2-carboxamide Authors: Longenecker, K.L, Bigelow, L. Deposit date: 2019-04-22 Release date: 2020-01-29 Last modified: 2024-03-13 Method: X-RAY DIFFRACTION (1.98 Å) Cite: Selective inhibition of the BD2 bromodomain of BET proteins in prostate cancer. Nature, 578, 2020

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2019-04-22
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