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Crystal Structure of Human p38alpha Complexed With a Triazolopyrimidine compound

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Protein Data Bank Japan2024-02-21 更新2026-03-21 收录
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Crystal Structure of Human p38alpha Complexed With a Triazolopyrimidine compound Descriptor: 3-{6-[2-(2,4-difluorophenyl)ethyl][1,2,4]triazolo[4,3-a]pyridin-3-yl}-4-methylbenzamide, Mitogen-activated protein kinase 14 Authors: Shieh, H.-S, Williams, J.M, Stegeman, R.A, Xing, L, Jerome, K.D. Deposit date: 2009-10-27 Release date: 2009-12-29 Last modified: 2024-02-21 Method: X-RAY DIFFRACTION (2 Å) Cite: Continued exploration of the triazolopyridine scaffold as a platform for p38 MAP kinase inhibition. Bioorg.Med.Chem.Lett., 20, 2010
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2009-10-27
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