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Kinase domain of cSrc in complex with RL104

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Protein Data Bank Japan2023-11-01 更新2026-03-21 收录
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资源简介:
Kinase domain of cSrc in complex with RL104 Descriptor: N-(4-{[4-({[1-(3-aminophenyl)-3-tert-butyl-1H-pyrazol-5-yl]carbamoyl}amino)phenyl]amino}quinazolin-6-yl)-3-(4-methylpiperazin-1-yl)propanamide, Proto-oncogene tyrosine-protein kinase Src Authors: Gruetter, C, Richters, A, Rauh, D. Deposit date: 2011-09-27 Release date: 2012-10-10 Last modified: 2023-11-01 Method: X-RAY DIFFRACTION (2.7 Å) Cite: Overcoming Gatekeeper Mutations in cSrc and Abl by Hybrid Compound Design To be Published
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2011-09-27
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