Structure of CDK9 in complex with cyclin T and a 2-amino-4-heteroaryl- pyrimidine inhibitor
收藏Protein Data Bank Japan2024-11-13 更新2026-03-21 收录
下载链接:
https://pdbj.org/mine/summary/4bci
下载链接
链接失效反馈官方服务:
资源简介:
Structure of CDK9 in complex with cyclin T and a 2-amino-4-heteroaryl- pyrimidine inhibitor Descriptor: 3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamide, CYCLIN-DEPENDENT KINASE 9, CYCLIN-T1 Authors: Hole, A.J, Baumli, S, Wang, S, Endicott, J.A, Noble, M.E.M. Deposit date: 2012-10-02 Release date: 2013-01-09 Last modified: 2024-11-13 Method: X-RAY DIFFRACTION (3.1 Å) Cite: Comparative Structural and Functional Studies of 4-(Thiazol- 5-Yl)-2-(Phenylamino)Pyrimidine-5-Carbonitrile Cdk9 Inhibitors Suggest the Basis for Isotype Selectivity. J.Med.Chem., 56, 2013
创建时间:
2012-10-02



