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PDK1 in complex with DFG-OUT inhibitor xxx

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Protein Data Bank Japan2024-10-16 更新2026-03-21 收录
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PDK1 in complex with DFG-OUT inhibitor xxx Descriptor: 1-(3,4-difluorobenzyl)-2-oxo-N-{(1R)-2-[(2-oxo-2,3-dihydro-1H-benzimidazol-5-yl)oxy]-1-phenylethyl}-1,2-dihydropyridine-3-carboxamide, 3-phosphoinositide-dependent protein kinase 1 Authors: Arndt, J.W. Deposit date: 2011-01-15 Release date: 2011-04-20 Last modified: 2024-10-16 Method: X-RAY DIFFRACTION (1.8 Å) Cite: Discovery of a potent and highly selective PDK1 inhibitor via fragment-based drug discovery. Bioorg.Med.Chem.Lett., 21, 2011

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2011-01-15
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