Crystal Structure of the first bromodomain of human BRD4 in complex with a quinazoline ligand
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Crystal Structure of the first bromodomain of human BRD4 in complex with a quinazoline ligand Descriptor: 1,2-ETHANEDIOL, Bromodomain-containing protein 4, N-ethyl-3-methyl-2-oxo-1,2,3,4-tetrahydroquinazoline-6-sulfonamide, ... Authors: Filippakopoulos, P, Picaud, S, Qi, J, Felletar, I, von Delft, F, Bountra, C, Arrowsmith, C.H, Edwards, A, Fish, P.V, Bunnage, M.E, Cook, A.S, Owen, D.R, Knapp, S, Structural Genomics Consortium (SGC) Deposit date: 2012-09-28 Release date: 2012-10-31 Last modified: 2023-09-20 Method: X-RAY DIFFRACTION (1.69 Å) Cite: Identification of a Chemical Probe for Bromo and Extra C-Terminal Bromodomain Inhibition through Optimization of a Fragment-Derived Hit. J.Med.Chem., 55, 2012
创建时间：
2012-09-28
