Crystal structure of C-terminal Domain of MSK1 in complex with covalently bound pyrrolopyrimidine compound 23 (co-crystal)
收藏Protein Data Bank Japan2024-11-13 更新2026-04-19 收录
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Crystal structure of C-terminal Domain of MSK1 in complex with covalently bound pyrrolopyrimidine compound 23 (co-crystal) Descriptor: (2M)-6-chloro-2-(5H-pyrrolo[3,2-d]pyrimidin-5-yl)pyridine-3-carbonitrile, IODIDE ION, Ribosomal protein S6 kinase alpha-5 Authors: Yano, J.K, Edwards, T.E, Hall, A. Deposit date: 2022-04-14 Release date: 2022-07-06 Last modified: 2024-11-13 Method: X-RAY DIFFRACTION (2.8 Å) Cite: Discovery and Characterization of a Novel Series of Chloropyrimidines as Covalent Inhibitors of the Kinase MSK1. Acs Med.Chem.Lett., 13, 2022
创建时间:
2022-04-14



