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Crystal structure of Lymnaea stagnalis Acetylcholine-binding protein (Ls-AChBP) Q55R/M114V double mutant complexed with Triflumezopyrim

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Protein Data Bank Japan2024-11-20 更新2026-05-23 收录
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Crystal structure of Lymnaea stagnalis Acetylcholine-binding protein (Ls-AChBP) Q55R/M114V double mutant complexed with Triflumezopyrim Descriptor: 4-oxidanylidene-1-(pyrimidin-5-ylmethyl)-3-[3-(trifluoromethyl)phenyl]pyrido[1,2-a]pyrimidin-1-ium-2-olate, Acetylcholine-binding protein Authors: Montgomery, M.G. Deposit date: 2021-08-09 Release date: 2022-02-02 Last modified: 2024-11-20 Method: X-RAY DIFFRACTION (2.1 Å) Cite: Structural Biology-Guided Design, Synthesis, and Biological Evaluation of Novel Insect Nicotinic Acetylcholine Receptor Orthosteric Modulators. J.Med.Chem., 65, 2022

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2021-08-09
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