Rip1 Kinase ( flag 1-294, C34A, C127A, C233A, C240A) with GSK772
收藏Protein Data Bank Japan2024-03-06 更新2026-03-21 收录
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https://pdbj.org/mine/summary/5tx5
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Rip1 Kinase ( flag 1-294, C34A, C127A, C233A, C240A) with GSK772 Descriptor: 3-benzyl-N-[(3S)-5-methyl-4-oxo-2,3,4,5-tetrahydro-1,5-benzoxazepin-3-yl]-1H-1,2,4-triazole-5-carboxamide, Receptor-interacting serine/threonine-protein kinase 1 Authors: Campobasso, N, Ward, P, Thrope, J. Deposit date: 2016-11-15 Release date: 2017-07-05 Last modified: 2024-03-06 Method: X-RAY DIFFRACTION (2.56 Å) Cite: Discovery of a First-in-Class Receptor Interacting Protein 1 (RIP1) Kinase Specific Clinical Candidate (GSK2982772) for the Treatment of Inflammatory Diseases. J. Med. Chem., 60, 2017
创建时间:
2016-11-15



