Human B-Raf Kinase in Complex with an Amide Linked Pyrazolopyridine Inhibitor
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Human B-Raf Kinase in Complex with an Amide Linked Pyrazolopyridine Inhibitor Descriptor: 2,6-difluoro-N-[(5S)-3-methoxy-5H-pyrazolo[3,4-b]pyridin-5-yl]-3-[(phenylsulfonyl)amino]benzamide, Serine/threonine-protein kinase B-raf Authors: Voegtli, W.C, Sturgis, H.L. Deposit date: 2011-06-22 Release date: 2011-08-17 Last modified: 2024-02-28 Method: X-RAY DIFFRACTION (3.2 Å) Cite: Pyrazolopyridine inhibitors of B-RafV600E. Part 2: structure-activity relationships. Bioorg.Med.Chem.Lett., 21, 2011
创建时间:
2011-06-22



