Mtb GuaB dCBS in complex with inhibitor G1
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Mtb GuaB dCBS in complex with inhibitor G1 Descriptor: INOSINIC ACID, Inosine-5'-monophosphate dehydrogenase, N-(6-chloropyridin-3-yl)-N~2~-(1,4-dihydro-2H-pyrano[3,4-c]quinolin-9-yl)-L-alaninamide, ... Authors: Harris, S.F, Wu, P. Deposit date: 2024-08-25 Release date: 2024-11-27 Last modified: 2025-01-29 Method: X-RAY DIFFRACTION (1.6 Å) Cite: Discovery of potent dihydro-oxazinoquinolinone inhibitors of GuaB for the treatment of tuberculosis. Bioorg.Med.Chem.Lett., 117, 2025
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2024-08-25



