Crystal Structure of Human BACE-1 in Complex with CNP520
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Crystal Structure of Human BACE-1 in Complex with CNP520 Descriptor: Beta-secretase 1, ~{N}-[6-[(3~{R},6~{R})-5-azanyl-3,6-dimethyl-6-(trifluoromethyl)-2~{H}-1,4-oxazin-3-yl]-5-fluoranyl-pyridin-2-yl]-3-chloranyl-5-(trifluoromethyl)pyridine-2-carboxamide Authors: Rondeau, J.-M, Wirth, E. Deposit date: 2017-10-13 Release date: 2018-09-19 Last modified: 2024-10-16 Method: X-RAY DIFFRACTION (1.35 Å) Cite: The BACE-1 inhibitor CNP520 for prevention trials in Alzheimer's disease. EMBO Mol Med, 10, 2018
创建时间:
2017-10-13



