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Crystal structure of human 3-phosphoglycerate dehydrogenase in complex with 3-Hydroxybenzisoxazole

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Protein Data Bank Japan2024-05-08 更新2026-03-21 收录
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Crystal structure of human 3-phosphoglycerate dehydrogenase in complex with 3-Hydroxybenzisoxazole Descriptor: 1,2-benzoxazol-3-ol, D-3-phosphoglycerate dehydrogenase Authors: Unterlass, J.E, Basle, A, Blackburn, T.J, Tucker, J, Cano, C, Noble, M.E.M, Curtin, N.J. Deposit date: 2017-05-14 Release date: 2017-06-14 Last modified: 2024-05-08 Method: X-RAY DIFFRACTION (1.3 Å) Cite: Validating and enabling phosphoglycerate dehydrogenase (PHGDH) as a target for fragment-based drug discovery in PHGDH-amplified breast cancer. Oncotarget, 9, 2018
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2017-05-14
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