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complex of human phosphoinositide 3-kinase catalytic subunit gamma (p110 gamma) with PIK-284

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Protein Data Bank Japan2023-12-13 更新2026-03-21 收录
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https://pdbj.org/mine/summary/2v4l
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资源简介:
complex of human phosphoinositide 3-kinase catalytic subunit gamma (p110 gamma) with PIK-284 Descriptor: 3-[4-AMINO-1-(1-METHYLETHYL)-1H-PYRAZOLO[3,4-D]PYRIMIDIN-3-YL]PHENOL, PHOSPHATIDYLINOSITOL-4,5-BISPHOSPHATE 3-KINASE CATALYTIC SUBUNIT GAMMA ISOFORM Authors: Apsel, B, Gonzalez, B, Blair, J.A, Nazif, T.M, Feldman, M.E, Williams, R.L, Shokat, K.M, Knight, Z.A. Deposit date: 2008-09-25 Release date: 2008-10-14 Last modified: 2023-12-13 Method: X-RAY DIFFRACTION (2.5 Å) Cite: Targeted Polypharmacology: Discovery of Dual Inhibitors of Tyrosine and Phosphoinositide Kinases. Nat.Chem.Biol., 4, 2008
创建时间:
2008-09-25
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