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Structure-Based Design of ASK1 Inhibitors as Potential First-in-Class Agents for Heart Failure

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Protein Data Bank Japan2024-03-06 更新2026-03-21 收录
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Structure-Based Design of ASK1 Inhibitors as Potential First-in-Class Agents for Heart Failure Descriptor: 6-{[(2S)-4-methylmorpholin-2-yl]methoxy}-2-{6-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]pyridin-2-yl}-2,3-dihydro-1H-isoindol-1-one, Mitogen-activated protein kinase kinase kinase 5, SULFATE ION Authors: Dougan, D.R. Deposit date: 2017-02-01 Release date: 2017-06-07 Last modified: 2024-03-06 Method: X-RAY DIFFRACTION (2.75 Å) Cite: Structure-Based Design of ASK1 Inhibitors as Potential Agents for Heart Failure. ACS Med Chem Lett, 8, 2017
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2017-02-01
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