Menin bound to inhibitor M-808
收藏Protein Data Bank Japan2023-10-18 更新2026-03-21 收录
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Menin bound to inhibitor M-808 Descriptor: Menin, methyl [(1S,2R)-2-{(1S)-2-(azetidin-1-yl)-1-(3-fluorophenyl)-1-[1-({1-[4-({1-[4-(piperidin-1-yl)butanoyl]azetidin-3-yl}sulfonyl)phenyl]azetidin-3-yl}methyl)piperidin-4-yl]ethyl}cyclopentyl]carbamate, praseodymium triacetate Authors: Stuckey, J.A. Deposit date: 2020-04-22 Release date: 2020-05-13 Last modified: 2023-10-18 Method: X-RAY DIFFRACTION (2.1 Å) Cite: Discovery of M-808 as a Highly Potent, Covalent, Small-Molecule Inhibitor of the Menin-MLL Interaction with StrongIn VivoAntitumor Activity. J.Med.Chem., 63, 2020
创建时间：
2020-04-22
