Fragment-based screening identifies a new area for inhibitor binding to checkpoint kinase 2 (CHK2)
收藏Protein Data Bank Japan2023-12-20 更新2026-03-21 收录
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Fragment-based screening identifies a new area for inhibitor binding to checkpoint kinase 2 (CHK2) Descriptor: 1,2-ETHANEDIOL, 1-acetyl-N-(5-methylpyridin-2-yl)piperidine-4-carboxamide, CHLORIDE ION, ... Authors: Silva-Santisteban, M.C, Westwood, I.M, Boxall, K, Brown, N, Peacock, S, McAndrew, C, Barrie, E, Richards, M, Mirza, A, Oliver, A.W, Burke, R, Hoelder, S, Jones, K, Aherne, G.W, Blagg, J, Collins, I, Garrett, M.D, van Montfort, R.L.M. Deposit date: 2012-10-05 Release date: 2013-06-26 Last modified: 2023-12-20 Method: X-RAY DIFFRACTION (2.32 Å) Cite: Fragment-Based Screening Maps Inhibitor Interactions in the ATP-Binding Site of Checkpoint Kinase 2. Plos One, 8, 2013
创建时间:
2012-10-05



