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CRYSTAL STRUCTURE OF HIV-1 V106A and Y181C MUTANT REVERSE TRANSCRIPTASE IN COMPLEX WITH GW564511.

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Protein Data Bank Japan2024-11-20 更新2026-03-21 收录
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CRYSTAL STRUCTURE OF HIV-1 V106A and Y181C MUTANT REVERSE TRANSCRIPTASE IN COMPLEX WITH GW564511. Descriptor: N-{4-[amino(dihydroxy)-lambda~4~-sulfanyl]-2-methylphenyl}-2-(4-chloro-2-{[3-fluoro-5-(trifluoromethyl)phenyl]carbonyl}phenoxy)acetamide, PHOSPHATE ION, Reverse transcriptase/ribonuclease H, ... Authors: Ren, J, Chamberlain, P.P, Stammers, D.K. Deposit date: 2008-07-01 Release date: 2008-08-12 Last modified: 2024-11-20 Method: X-RAY DIFFRACTION (2.6 Å) Cite: Structural basis for the improved drug resistance profile of new generation benzophenone non-nucleoside HIV-1 reverse transcriptase inhibitors. J.Med.Chem., 51, 2008
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2008-07-01
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